Naloxonazine dihydrochloride
Cat. No.:YN322683
产品名称: | Naloxonazine dihydrochloride |
CAS No.: | 880759-65-9 |
Chemical Name: | (5α)-[(5α)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazone, 4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)-morphinan-6-one, dihydrochloride |
Synonyms: | |
分子量: | 723.7 |
分子式: | C38H42N4O6 • 2HCl |
SMILES: | O[C@]12[C@]3(CCN(CC=C)[C@@H]2C4)[C@](OC5=C3C4=CC=C5O)([H])/C(CC1)=N/N=C(CC[C@@]6(O)[C@H]7CC8=CC=C9O)/[C@@]%10([H])[C@]6(CCN7CC=C)C8=C9O%10.Cl.Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Naloxonazine dihydrochloride 是一种特异性的μ-opioid receptor拮抗剂,IC50为 5.4 nM。Naloxonazine dihydrochloride 也具有抗利什曼原虫活性。 |
IC50和靶点: | [{name:"μ Opioid Receptor/MOR:5.4 nM (IC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
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