Velusetrag
Cat. No.:YN322800
产品名称: | Velusetrag |
CAS No.: | 866933-46-2 |
Chemical Name: | |
Synonyms: | TD-5108 |
分子量: | 504.646 |
分子式: | C25H36N4O5S |
SMILES: | CN(C[C@H](O)CN1C2CC(NC(=O)C3C(=O)N(C(C)C)C4C(=CC=CC=4)C=3)CC1CC2)S(=O)(C)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Velusetrag (TD-5108) 是一种具有口服活性,有效和选择性的血清素5-HT4受体 (5-HT4R) 激动剂,pKi为 7.7。Velusetrag 对 5-HT2A和 5-HT2B受体没有亲和力 (Ki>10 μM)。Velusetrag 可用于胃肠道疾病和帕金森病的研究。 |
IC50和靶点: | [{name:"5-HT4 Receptor:7.7 (pKi)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |