S-777469
Cat. No.:YN322802
产品名称: | S-777469 |
CAS No.: | 885496-53-7 |
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分子量: | 414.47 |
分子式: | C23H27FN4O2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | S-777469 是一种选择性,具有口服活性的大麻素 2 型受体(CB2)激动剂,Ki为 36 nM。S-777469 以剂量依赖性方式显著抑制化合物 48/80 诱导的小鼠抓挠行为。S-777469 通过CB2兴奋抑制瘙痒信号的传递,从而产生止痒作用。 |
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