Pitofenone hydrochloride
Cat. No.:YN380041
CAS No. :1248-42-6
产品名称: | Pitofenone hydrochloride |
CAS No.: | 1248-42-6 |
Chemical Name: | 2-[4-[2-(1-piperidinyl)ethoxy]benzoyl]-benzoic acid, methyl ester, monohydrochloride |
Synonyms: | Baralgin Ketone Hydrochloride,Pitophenone hydrochloride,吡托非农盐酸盐 |
分子量: | 403.90 |
分子式: | C₂₂H₂₆ClNO₄ |
SMILES: | Cl[H].O=C(C1=CC=C(C=C1)OCCN2CCCCC2)C3=C(C=CC=C3)C(OC)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Pitofenone hydrochloride 是一种解痉化合物,能够抑制乙酰胆碱酯酶 (AChE) 的活性,对于来自牛红细胞和电鳗的乙酰胆碱酯酶的Ki值分别为 36 和 45 μM。 |
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Punekar, N.S., and Kulkarni, A.V.Acetylcholinesterase inhibition by pitofenone: A spasmolytic compoundBiotechnol. Appl. Biochem.14(3),378-382(1991)
Kulkarni, S.K., Patil, C.S., and Singh, A.Modulatory effect of diclofenac on antispasmodic effect of pitofenone in cholinergic spasmIndian J. Exp. Biol.42(6),567-569(2004)