ALK-IN-1
Cat. No.:YN440273
产品名称: | ALK-IN-1 |
CAS No.: | 1197958-12-5 |
Chemical Name: | 5-chloro-N2-[4-[4-(dimethylamino)-1-piperidinyl]-2-methoxyphenyl]-N4-[2-(dimethylphosphinyl)phenyl]-2,4-pyrimidinediamine |
Synonyms: | Brigatinib analog |
分子量: | 529.01 |
分子式: | C₂₆H₃₄ClN₆O₂P |
SMILES: | CP(C)(C1=CC=CC=C1NC2=NC(NC3=CC=C(N4CCC(N(C)C)CC4)C=C3OC)=NC=C2Cl)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | ALK-IN-1 (Brigatinib analog) 是ALK激酶高效选择性抑制剂,出自专利 US20140066406 A1。 |
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Huang, W.S., Liu, S., Zou, D., et al.Discovery of brigatinib (AP26113), a phosphine oxide-containing, potent, orally active inhibitor of anaplastic lymphoma kinaseJ. Med. Chem.,(2016)