LUF6000
Cat. No.:YN1570003
CAS No. :890087-21-5
产品名称: | LUF6000 |
CAS No.: | 890087-21-5 |
Chemical Name: | 2-cyclohexyl-N-(3,4-dichlorophenyl)-3H-imidazo[4,5-c]quinolin-4-amine |
Synonyms: | LUF-6000;LUF 6000 |
分子量: | 411.33 |
分子式: | C₂₂H₂₀Cl₂N₄ |
SMILES: | ClC1=CC(NC2=NC3=C(C=CC=C3)C4=C2NC(C5CCCCC5)=N4)=CC=C1Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | LUF6000 是一种口服活性的 A3 腺苷受体 (A3 adenosine receptor) 的变构调节剂。LUF6000 具有强大的抗炎作用。 |
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Göblyös, A., Gao, Z.-G., Brussee, J., et al.Structure-activity relationships of new 1H-imidazo[4,5-c]quinolin-4-amine derivatives as allosteric enhancers of the A3 adenosine receptorJ. Med. Chem.49(11),3354-3361(2006)
Cohen, S., Barer, F., Bar-Yehuda, S., et al.A3 adenosine receptor allosteric modulator induces an anti-inflammatory effect: In vivo studies and molecular mechanism of actionMediators Inflamm.2014:708746,(2014)