MRS-1191
Cat. No.：YN1730047
CAS No. ：185222-90-6
| 产品名称: | MRS-1191 |
| CAS No.: | 185222-90-6 |
| Chemical Name: | 3-Ethyl 5-(phenylmethyl)-1,4-dihydro-2-methyl-6-phenyl-4-(phenylethynyl)-3,5-Pyridinedicarboxylic Acid Ester; |
| Synonyms: | MRS1191; MRS 1191; MRS-1191. |
| 分子量: | 477.55 |
| 分子式: | C₃₁H₂₇NO₄ |
| SMILES: | O=C(OCC)C1=C(NC(C2=CC=CC=C2)=C(C1C#CC3=CC=CC=C3)C(OCC4=CC=CC=C4)=O)C |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | MRS-1191 是一种有效的选择性的 A3腺苷受体 (A3adenosine receptor) 拮抗剂，其KB值为 92 nM，对人 A3受体的Ki值为 31.4 nM，对 CHO 细胞的IC50值为 120 nM。 |
| IC50和靶点: | |
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| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Jiang, J., et al.: J. Med. Chem., 39, 4667-4675 (1996)
Yao, Y., et al.: Biochem. Biophys. Res. Commun., 232, 317-322 (1997)
