Cimaterol-D7
Cat. No.:YN320089
CAS No. :1228182-44-2
产品名称: | Cimaterol-D7 |
CAS No.: | 1228182-44-2 |
Chemical Name: | 2-amino-5-[1-hydroxy-2-[[1-(methyl-d3)ethyl-1,2,2,2-d4]amino]ethyl]-benzonitrile |
Synonyms: | |
分子量: | 226.33 |
分子式: | C₁₂H₁₀D₇N₃O |
SMILES: | N#CC1=CC(C(O)CNC(C([2H])([2H])[2H])([2H])C([2H])([2H])[2H])=CC=C1N |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Cimaterol-D7 is the deuterium labeled Cimaterol. Cimaterol is a potent agonist of β-adrenergic receptors (pEC50s=8.13, 8.78, and 6.62 for human β1, β2, and β3, respectively). Cimaterol has been used in farmed animals to increase carcass mass and to alter |
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Mistry, S.N., Baker, J.G., Fischer, P.M., et al.Synthesis and in vitro and in vivo characterization of highly β1-selective β-adrenoceptor partial agonistsJ. Med. Chem.56(10),3852-3865(2013)
Jones, R.W., Easter, R.A., McKeith, F.K., et al.Effect of the β-adrenergic agonist cimaterol (CL 263,780) on the growth and carcass characteristics of finishing swineJ. Anim. Sci.61(4),905-913(1985)
Byrem, T.M., Beermann, D.H., and Robinson, T.F.The β-agonist cimaterol directly enhances chronic protein accretion in skeletal muscleJ. Anim. Sci.76(4),988-998(1998)