Salmeterol
Cat. No.:YN320848
CAS No. :89365-50-4
产品名称: | Salmeterol |
CAS No.: | 89365-50-4 |
Chemical Name: | (±)-4-Hydroxy-α1-[[[6-(4-phenylbutoxy)hexyl]amino]methyl]-1,3-benzenedimethanol; GR 33343X |
Synonyms: | 沙美特罗; GR33343X |
分子量: | 415.57 |
分子式: | C₂₅H₃₇NO₄ |
SMILES: | OC1=CC=C(C(O)CNCCCCCCOCCCCC2=CC=CC=C2)C=C1CO |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Salmeterol (GR33343X) 是长效β2肾上腺素受体激动剂,可作用于哮喘。 |
IC50和靶点: | [{name:"β2 adrenoceptor:9.6 (pEC50)"},{name: "β1 adrenoceptor:6.1 (pEC50)"},{name: "β3 adrenoceptor:5.9 (pEC50)"}] |
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Ullman, A., et al.: Am. Rev. Resp. Dis., 142, 571 (1990)
Twentyman, O.P., et al.: Lancet, 336, 1338 (1990)