Idazoxan hydrochloride
Cat. No.:YN320891
产品名称: | Idazoxan hydrochloride |
CAS No.: | 79944-56-2 |
Chemical Name: | 2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole Hydrochloride; (+/-)-Idazoxan Monohydrochloride; RX 781094; RX 781094A; |
Synonyms: | RX 781094 hydrochloride |
分子量: | 240.69 |
分子式: | C₁₁H₁₃ClN₂O₂ |
SMILES: | [H]Cl.C1(C2OC3=CC=CC=C3OC2)=NCCN1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Idazoxan hydrochloride (RX 781094 hydrochloride) 是一种 α2-肾上腺素受体拮抗剂,也是咪唑啉受体 (IRs) 拮抗剂,可竞争性拮抗唑啉样药物 (IMs) 的中枢性降压作用。Idazoxan hydrochloride 还可改善帕金森氏病,L-DOPA 引起的运动障碍和实验性帕金森病的运动症状。 |
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Fliri, A., et al.: Med. Chem., 48, 6918 (2005), Yildirim, M., et al.: Nat. Biotechnol., 25, 1119 (2007),