Fiduxosin
Cat. No.:YN322085
CAS No. :208993-54-8
产品名称: | Fiduxosin |
CAS No.: | 208993-54-8 |
Chemical Name: | 8-Phenyl-3-[4-[(3aR,9bR)-1,3a,4,9b-tetrahydro-9-methoxy[1]benzopyrano[3,4-c]pyrrol-2(3H)-yl]butyl]-pyrazino[2',3':4,5]thieno[3,2-d]pyrimidine-2,4(1H,3H)-dione; 3-(4-((3aR,9bR)-9-Methoxy-1,3a,4,9b-tetrahydrochromeno[3,4-c]pyrrol-2(3H)-yl)butyl)-8-phenylpyr |
Synonyms: | |
分子量: | 555.65 |
分子式: | C₃₀H₂₉N₅O₄S |
SMILES: | O=C(N1CCCCN2C[C@]3([H])[C@](COC4=CC=CC(OC)=C34)([H])C2)C5=C(NC1=O)C6=NC(C7=CC=CC=C7)=CN=C6S5 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Fiduxosin 是一种α1-adrenoceptor拮抗剂,对 α1a-adrenoceptor,α1b-adrenoceptor 和 α1d-adrenoceptor 的Ki值分别为 0.160 nM,24.9 nM 和 0.920 nM。 |
IC50和靶点: | |
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Clinical Trial: | |
Solvent & Solubility: |
Dutta, S., et. al.: J. Pharm. Pharm., 54, 641 (2002)
Pan, P., Lu, J.: Zhongguo Yaoxue Zzhi, 41, 1521 (2006)