CGP-42112
Cat. No.:YN320590
产品名称: | CGP-42112 |
CAS No.: | 127060-75-7 |
Chemical Name: | N-(3-pyridinylcarbonyl)-L-tyrosyl-N6-[N2-[(phenylmethoxy)carbonyl]-L-arginyl]-L-lysyl-L-histidyl-L-prolyl-L-isoleucine |
Synonyms: | CGP42112A |
分子量: | 1052.19 |
分子式: | C₅₂H₆₉N₁₃O₁₁ |
SMILES: | CC[C@H](C)[C@@H](C(O)=O)NC([C@H]1N(C([C@H](CC2=CNC=N2)NC([C@H](CCCCNC([C@H](CCCNC(N)=N)NC(OCC3=CC=CC=C3)=O)=O)NC([C@H](CC4=CC=C(C=C4)O)NC(C5=CC=CN=C5)=O)=O)=O)=O)CCC1)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CGP-42112(CGP-42112A)是血管紧张素受体AT2激动剂。 |
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Criscione, L., Thomann, H., Whitebread, S., et al.Binding characteristics and vascular effects of various angiotensin II antagonistsJ. Cardiovasc. Pharmacol.16 (Suppl 4),S56-S59(1990)
Takekoshi, K., Isobe, K.I., Nanmoku, T., et al.Angiotensin-II subtype 2 receptor agonist (CGP-42112) inhibits catecholamine biosynthesis in cultured porcine adrenal medullary chromaffin cellsBiochem. Biophys. Res. Commun.272(2),544-550(2000)