Quinidine gluconic acid
Cat. No.：YN252017
| 产品名称: | Quinidine gluconic acid |
| CAS No.: | 126062-19-9 |
| Chemical Name: | 7-amino-4-chloro-3-propoxy-1H-2-benzopyran-1-one |
| Synonyms: | 1H-2-Benzopyran-1-one, 7-amino-4-chloro-3-propoxy-;7-Amino-4-chloro-3-propoxy-isochromen-1-one |
| 分子量: | 253.7 |
| 分子式: | C12H12ClNO3 |
| SMILES: | NC1=CC=C2C(C(OC(OCCC)=C2Cl)=O)=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | JCP174 是棕榈酰蛋白硫酯酶-1 (TgPPT1) 的抑制剂，该酶是弓形虫体内的一种去棕榈酰化酶。JCP174 也是猪胰腺弹性蛋白酶和人类白细胞弹性蛋白酶的抑制剂。 |
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Kerrigan, J.E., Oleksyszyn, J., Kam, C.-M., et al.Mechanism-based isocoumarin inhibitors for human leukocyte elastase. Effect of the 7-amino substituent and 3-alkoxy group in 3-alkoxy-7-amino-4-chloroisocoumarins on inhibitory potencyJ. Med. Chem.38(3),544-552(1995)
