Chrysomycin A
Cat. No.:YN252323
产品名称: | Chrysomycin A |
CAS No.: | 739-71-9 |
Chemical Name: | |
Synonyms: | 曲米帕明 |
分子量: | 暂无 |
分子式: | 暂无 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Trimipramine 是5-HT受体的拮抗剂,其对 5-HT1C,5-HT2和 5-HT1A受体的 pKi值分别为 6.39,8.10,4.66。Trimipramine 也是一种靶向人去甲肾上腺素 (hNAT)、血清素 (hSERT) 和有机阳离子转运体 (hOCT1、hOCT2) 的有选择性和强效的抑制剂,其IC50值分别为 4.99 μM、2.11 μM、3.72 μM、8.00 μM。Trimipramine 具有血管活性和抗焦虑作用。 |
IC50和靶点: | [{name:"5-HT1C Receptor:6.39 (pKi)"},{name: "5-HT2 Receptor:8.10 (pKi)"},{name: "5-HT1A Receptor:4.66 (pKi)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |