α-NETA
Cat. No.:YN270179
CAS No. :31059-54-8
产品名称: | α-NETA |
CAS No.: | 31059-54-8 |
Chemical Name: | N,N,N-trimethyl-γ-oxo-2-naphthalenepropanaminium, monoiodide |
Synonyms: | α-NETA |
分子量: | 369.24 |
分子式: | C₁₆H₂₀INO |
SMILES: | O=C(C1=CC=C2C=CC=CC2=C1)CC[N+](C)(C)C.[I-] |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | α-NETA 是一种稳定的,非竞争性的,缓慢可逆的胆碱乙酰转移酶 (ChAT) 抑制剂,IC50为 9 μM。α-NETA 是一种有效的趋化因子样受体1 (CMKLR1) 拮抗剂。α-NETA 微弱的抑制胆碱酯酶(IC50= 84 µM)和乙酰胆碱酯(IC50= 300 µM)。α-NETA 具有抗癌活性。 |
IC50和靶点: | |
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