Tasisulam
Cat. No.:YN270291
CAS No. :519055-62-0
产品名称: | Tasisulam |
CAS No.: | 519055-62-0 |
Chemical Name: | N-[(5-bromo-2-thienyl)sulfonyl]-2,4-dichloro-benzamide |
Synonyms: | LY 573636 |
分子量: | 415.11 |
分子式: | C₁₁H₆BrCl₂NO₃S₂ |
SMILES: | O=C(NS(=O)(C1=CC=C(Br)S1)=O)C2=CC=C(Cl)C=C2Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Tasisulam 是一种小分子抗肿瘤药物,通过内在途径诱导细胞凋亡,导致细胞色素 c 释放和 caspase 依赖性细胞死亡。Tasisulam 可以抑制有丝分裂进程并诱导血管正常化。 |
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Meier, T., Uhlik, M., Chintharlapalli, S., et al.Tasisulam sodium, an antitumor agent that inhibits mitotic progression and induces vascular normalizationMol. Cancer. Ther.10(11),2168-2178(2011)