(Rac)-Rotigotine-d
Cat. No.:YN322159
产品名称: | (Rac)-Rotigotine-d |
CAS No.: | 1126745-58-1 |
Chemical Name: | 5-[2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl-2,2,3,3,5,5,6,6-d8]ethyl]-6-chloro-1,3-dihydro-2H-indol-2-one |
Synonyms: | 齐哌西酮D8; CP-88059 d |
分子量: | 420.98498 |
分子式: | C21H13D8ClN4OS |
SMILES: | [2H]C(C([2H])([2H])N(CCC1=C(Cl)C=C(NC(C2)=O)C2=C1)C([2H])([2H])C3([2H])[2H])([2H])N3C4=NSC5=CC=CC=C54 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Ziprasidone-d88是Ziprasidone的氘代标记化合物。 |
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Seeman, P.Atypical antipsychotics: Mechanism of actionCan. J. Psychiatry47(1),27-38(2002)
Schmidt, A.W., Lebel, L.A., Howard, H.R., Jr., et al.Ziprasidone: A novel antipsychotic agent with a unique human receptor binding profileEur. J. Pharmacol.425(3),197-201(2001)
Audinot, V., Newman-Tancredi, A., Cussac, D., et al.Inverse agonist properties of antipsychotic agents at cloned, human (h) serotonin (5-HT)1B and h5-HT1D receptorsNeuropsychopharmacology25(3),410-422(2001)
Seeger, T.F., Seymour, P.A., Schmidt, A.W., et al.Ziprasidone (CP-88,059): A new antipsychotic with combined dopamine and serotonin receptor antagonist activityJ. Pharmacol. Exp. Ther.275(1),101-113(1995)