Artemisitene
Cat. No.:YN290560
产品名称: | Artemisitene |
CAS No.: | 101020-89-7 |
Chemical Name: | (3R,5aS,6R,8aS,12S,12aR)-Octahydro-3,6-dimethyl-9-methylene-3,12-epoxy-12H-pyrano[4,3-j]-1,2-benzodioxepin-10(3H)-one; (+)-Artemisitene; Dehydroqinghaosu; |
Synonyms: | 青蒿烯 |
分子量: | 280.316305160522 |
分子式: | C15H20O5 |
SMILES: | O=C1O[C@H]2[C@@]34OO[C@](O2)(C)CC[C@H]3[C@@H](CC[C@H]4C1=C)C |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Artemisitene 是 Artemisinin 的天然衍生物,是一种Nrf2激活剂,具有抗氧化和抗癌活性。Artemisitene 通过降低 Nrf2 泛素化并增加其稳定性来激活 Nrf2。 |
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Li, Y., et al.: Curr. Med. Chem., 10, 2197 (2003), Marrero-Ponce, Y., et al.: Bioorg. Med. Chem., 13, 1293 (2005), McMichael, A., et al.: Lancet, 367, 859 (2006),