BRD4-IN-3
Cat. No.：YN310415
| 产品名称: | BRD4-IN-3 |
| CAS No.: | 1380087-86-4 |
| Chemical Name: | (4S)-8-chloro-6-(4-chlorophenyl)-1-methyl-4H-isoxazolo[5,4-d][2]benzazepine-4-acetamide |
| Synonyms: | CPI-268456 |
| 分子量: | 400.3 |
| 分子式: | C20H15Cl2N3O2 |
| SMILES: | NC(C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C3=C(C=CC(Cl)=C3)C4=C1ON=C4C)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | BRD4-IN-3 (compound 141) 是一种有效的BRD4抑制剂，IC50为 <0.5 µM。BRD4-IN-3 对 MYC-Raji 显示细胞毒性，IC50值 >1 µM。 |
| IC50和靶点: | [{name:"BRD4:<0.5 μM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Albrecht, B.K., Audia, J.E., Côté, A., et al.Bromodomain inhibitors and uses thereof,(2012)
