I-BET282
Cat. No.:YN310419
CAS No. :1422554-34-4
产品名称: | I-BET282 |
CAS No.: | 1422554-34-4 |
Chemical Name: | |
Synonyms: | |
分子量: | 450.53 |
分子式: | C25H30N4O4 |
SMILES: | COC1=C(C2=C(C)ON=C2C)C=C(N=CC3=C4N(C(C5CCOCC5)=N3)[C@@H](COC)C)C4=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | I-BET282 是八种BET bromodomains泛抑制剂,对其他代表性含溴代烷的蛋白质具有选择性。I-BET282 对 8 种BRD2(BD1/BD2),BRD2(BD1/BD),BRD3(BD1/BD),BRD4(BD1/BD) 的 pIC50值为 6.4-7.7。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |