Bizine
Cat. No.:YN310431
产品名称: | Bizine |
CAS No.: | 1591932-50-1 |
Chemical Name: | N-[4-(2-hydrazinylethyl)phenyl]-benzenebutanamide |
Synonyms: | |
分子量: | 297.4 |
分子式: | C18H23N3O |
SMILES: | NNCCC(C=C1)=CC=C1NC(CCCC2=CC=CC=C2)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Bizine 是一种 Phenelzine 类似物,是有效和选择性的LSD1抑制剂,Ki值为 59 nM。Bizine 可以调节癌细胞中的组蛋白甲基化。Bizine 显示出神经保护作用。 |
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Prusevich, P., Kalin, J.H., Ming, S.A., et al.A selective phenelzine analogue inhibitor of histone demethylase LSD1ACS Chem Biol.9,1284-1293(2014)