GS-626510
Cat. No.：YN310433
CAS No. ：1637770-13-8
| 产品名称: | GS-626510 |
| CAS No.: | 1637770-13-8 |
| Chemical Name: | |
| Synonyms: | GS-6510;GS 6510;GS 626510 |
| 分子量: | 394.47 |
| 分子式: | C25H22N4O |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | GS-626510 是一个有效的、且具有口服活性的BET家族的抑制剂，其对 BRD2/3/4 的Kd值为 0.59-3.2 nM，对BD1和BD2的IC50值分别为 83 nM 和78 nM。 |
| IC50和靶点: | [{name:"BRD2:0.59-2.5 nM (Kd)"},{name: "BRD3:0.65-0.66 nM (Kd)"},{name: "BRD4:1.3-3.2 nM (Kd)"},{name: "BD1:83 nM (IC50)"},{name: "BD2:78 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
