Valemetostat
Cat. No.：YN310442
| 产品名称: | Valemetostat |
| CAS No.: | 1809336-39-7 |
| Chemical Name: | (2R)-7-chloro-N-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-2-[trans-4-(dimethylamino)cyclohexyl]-2,4-dimethyl-1,3-benzodioxole-5-carboxamide |
| Synonyms: | DS-3201 |
| 分子量: | 488.01868 |
| 分子式: | C26H34ClN3O4 |
| SMILES: | CC1=C2C(O[C@@](O2)([C@]3([H])CC[C@H](CC3)N(C)C)C)=C(C=C1C(NCC4=C(C=C(NC4=O)C)C)=O)Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Valemetostat (DS-3201) 是一种首创的EZH1/2抑制剂，IC50值 ＜10 nM。Valemetostat 可用于复发以及难治型周围 T 细胞淋巴瘤的研究。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
Honma, D., Kanno, O., Watanabe, J., et al.Novel orally bioavailable EZH1/2 dual inhibitors with greater antitumor efficacy than an EZH2 selective inhibitorCancer Sci.108(10),2069-2078(2017)
