GSK8814
Cat. No.：YN310457
| 产品名称: | GSK8814 |
| CAS No.: | 1997369-78-4 |
| Chemical Name: | |
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| 分子量: | 527.61 |
| 分子式: | C28H35F2N5O3 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | GSK8814 是一种高效、选择性的ATAD2/2B溴代苯胺化学探针和抑制剂，结合常数pKd=8.1，在 BROMOscan 中的pKi=8.9。GSK8814 分别以 7.3 和 4.6 的pIC50与 ATAD2 和BRD4BD1 结合。GSK8814 对 ATAD2 的选择性是BRD4BD1 的 500 倍。 |
| IC50和靶点: | [{name:"ATAD2:8.9 (pKi)"},{name: "ATAD2:8 nM (Ki)"},{name: "BRD4 BD1:4.6 (pIC50)"}] |
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