SR 16832
Cat. No.:YN290678
产品名称: | SR 16832 |
CAS No.: | 2088135-12-8 |
Chemical Name: | 2-chloro-N-(6-methoxy-4-quinolinyl)-5-nitro-benzamide |
Synonyms: | 2-chloro-N-(6-methoxy-4-quinolinyl)-5-nitro-benzamide |
分子量: | 357.7477 |
分子式: | C17H12ClN3O4 |
SMILES: | COC1=CC=C2C(C(NC(C3=CC([N+]([O-])=O)=CC=C3Cl)=O)=CC=N2)=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | SR 16832 是一种双位点共价的PPARγ抑制剂,作用于正构和变构位点。 |
IC50和靶点: | |
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Brust, R., Lin, H., Fuhrmann, J., et al.Modification of the orthosteric PPARγ covalent antagonist scaffold yields an improved dual-site allosteric inhibitorACS Chem. Biol.12(4),969-978(2017)