CPI-455 hydrochloride
Cat. No.:YN310465
产品名称: | CPI-455 hydrochloride |
CAS No.: | 2095432-28-1 |
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分子量: | 314.77 |
分子式: | C16H15ClN4O |
SMILES: | CC(C)C1=C(N=C2C(=CNN2C1=O)C#N)C3=CC=CC=C3.Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CPI-455 hydrochloride 是一种特异性的泛KDM5抑制剂,对 KDM5A 的IC50为 10 nM,CPI-455 hydrochloride 介导KDM5抑制,提高 H3K4me3 的整体水平,并减少多肿瘤细胞系模型中耐药的持久癌细胞的数量。 |
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