dCBP-1
Cat. No.:YN310497
CAS No. :2484739-25-3
产品名称: | dCBP-1 |
CAS No.: | 2484739-25-3 |
Chemical Name: | |
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分子量: | 1028.11 |
分子式: | C51H63F2N11O10 |
SMILES: | CNC(=O)N1CCC2=C(C1)C(=N[N]2C3CCN(CC3)C(=O)CCOCCOCCOCCOCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)N7CCCC8=CC(=C(C=C78)C(F)F)C9=C[N](C)N=C9 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | dCBP-1 是一种基于Cereblon配体的p300/CBP的有效且选择性的异双功能降解剂。dCBP-1 在杀死多发性骨髓瘤细胞方面非常有效,并降低了驱动 MYC 表达的致癌增强子活性。 |
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