H-Trp-Glu-OH
Cat. No.：YN290764
| 产品名称: | H-Trp-Glu-OH |
| CAS No.: | 36099-95-3 |
| Chemical Name: | L-tryptophyl-L-glutamic acid |
| Synonyms: | G3335 |
| 分子量: | 333.3 |
| 分子式: | C16H19N3O5 |
| SMILES: | OC(CC[C@@H](C(O)=O)NC([C@@H](N)CC1=CNC2=C1C=CC=C2)=O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | H-Trp-Glu-OH 是一种选择性的、可逆的且有细胞通透性的PPARγ拮抗剂，其Kd约为 8 µM。H-Trp-Glu-OH 可能作为研究糖尿病的先导化合物。 |
| IC50和靶点: | [{name:"PPARγ:8 μM (Kd)"}] |
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Ye, F., Zhang, Z.S., Luo, H.B., et al.The dipeptide H-Trp-Glu-OH shows highly antagonistic activity against PPARγ: Bioassay with molecular modeling simulationChembiochem7,74-82(2006)
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