ML192
Cat. No.:YN310514
CAS No. :460331-61-7
产品名称: | ML192 |
CAS No.: | 460331-61-7 |
Chemical Name: | 2-furanyl[4-(5,6,7,8-tetrahydro-2-methyl[1]benzothieno[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-methanone |
Synonyms: | ML192; ML 192; ML-192; CID1434953; CID-1434953; CID 1434953; MLS000526305. |
分子量: | 382.5 |
分子式: | C20H22N4O2S |
SMILES: | O=C(C1=CC=CO1)N2CCN(C3=C4C(SC5=C4CCCC5)=NC(C)=N3)CC2 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | ML192 是一种选择性的GPR55配体拮抗剂。ML192 抑制β-arrestin转运、ERK1/2磷酸化和PKCβII易位。 |
IC50和靶点: | |
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Solvent & Solubility: |
Heynen-Genel, S., Dahl, R., Shi, S., et al.Selective GPR55 antagonists: Screening for selective ligands for GPR55Probe Reports from the NIH Molecular Libraries Program,(2011)