HDAC/BET-IN-1
Cat. No.：YN290814
| 产品名称: | HDAC/BET-IN-1 |
| CAS No.: | 847459-98-7 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 456.92 |
| 分子式: | C23H25ClN4O4 |
| SMILES: | O=C(C(N1)=CC2=C1C=CC(OCCN(C)C)=C2)NCC#CC3=CC=C(C(NO)=O)C=C3.[H]Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | CRA-026440 hydrochloride 是一种有效的广谱HDAC(HDAC) 抑制剂。作用于HDAC1，HDAC2，HDAC3，HDAC6，HDAC8和HDAC10的Ki分别为 4 nM，14 nM，11 nM，15 nM，7 nM 和 20 nM。CRA-026440 hydrochloride 具有抗肿瘤和抗血管生成活性。 |
| IC50和靶点: | [{name:"HDAC1:4 nM (IC50)"},{name: "HDAC2:14 nM (IC50)"},{name: "HDAC3/SMRT:11 nM (IC50)"},{name: "HDAC6:15 nM (IC50)"},{name: "HDAC8:7 nM (IC50)"},{name: "HDAC10:20 nM (IC50)"}] |
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