FT-001
Cat. No.:YN310573
CAS No. :1778655-51-8
产品名称: | FT-001 |
CAS No.: | 1778655-51-8 |
Chemical Name: | |
Synonyms: | (S)-1-(4-(cyclopropanecarbonyl)-6-(4-(1,1-dioxidothiomorpholino)phenyl)-2-methyl-3,4-dihydroquinoxalin-1(2H)-yl)ethan-1-one |
分子量: | 467.584 |
分子式: | C25H29N3O4S |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | FT001是一种有效的、选择性的和具有口服活性的 BET Bromodomain抑制剂,具有抗肿瘤活性。FT001抑制MYC的表达,IC50为0.46 μM。FT001对MV-4-11具有有效的抗增殖作用,并在体外和体内显著抑制MYC mRNA水平。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |