N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(N-ethylcyclopropanecarboxamido)-4-methyl-4′-morpholino-[1,1′-biphenyl]-3-carboxamide
Cat. No.:YN310586
CAS No. :2238820-26-1
产品名称: | N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(N-ethylcyclopropanecarboxamido)-4-methyl-4′-morpholino-[1,1′-biphenyl]-3-carboxamide |
CAS No.: | 2238820-26-1 |
Chemical Name: | |
Synonyms: | |
分子量: | 542.68 |
分子式: | C32H38N4O4 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(N-ethylcyclopropanecarboxamido)-4-methyl-4′-morpholino-[1,1′-biphenyl]-3-carboxamide是一种强效的、选择性的Enhancer of Zeste Homolog 2 (EZH2),对EZH2 WT和EZH2-Y641F的IC50分别为37.6nM和79.1nM。 |
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