CCT020312
Cat. No.:YN280031
产品名称: | CCT020312 |
CAS No.: | 324759-76-4 |
Chemical Name: | 6-bromo-3-[5-(4-bromophenyl)-1-[3-(diethylamino)-1-oxopropyl]-4,5-dihydro-1H-pyrazol-3-yl]-4-phenyl-2(1H)-quinolinone |
Synonyms: | |
分子量: | 650.40 |
分子式: | C₃₁H₃₀Br₂N₄O₂ |
SMILES: | O=C1NC2=C(C(C3=CC=CC=C3)=C1C4=NN(C(C4)C5=CC=C(C=C5)Br)C(CCN(CC)CC)=O)C=C(C=C2)Br |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CCT020312 是选择性的EIF2AK3/PERK的激活剂。CCT020312 可诱导细胞细胞中 EIF2A 的磷酸化。 |
IC50和靶点: | |
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Solvent & Solubility: |
Stockwell, S.R., Platt, G., Barrie, S.E., et al.Mechanism-based screen for G1/S checkpoint activators identifies a selective activator of EIF2AK3/PERK signallingPLoS One7(1),e28568(2012)