Cilastatin sodium
Cat. No.:YN250877
CAS No. :81129-83-1
产品名称: | Cilastatin sodium |
CAS No.: | 81129-83-1 |
Chemical Name: | Cilastatin Sodium Salt; L 642957; MK 791; [R-[R*,S*-(Z)]]-7-[(2-Amino-2-carboxyethyl)thio]-2-[[(2,2-dimethylcyclopropyl)carbonyl]amino]-2-heptenoic Acid Monosodium Salt; (2Z)-7-[[(2R)-2-Amino-2-carboxyethyl]thio]-2-[[[(1S)-2,2-dimethylcyclo |
Synonyms: | 西司他丁钠; MK0791 sodium |
分子量: | 380.43 |
分子式: | C₁₆H₂₅N₂NaO₅S |
SMILES: | O=C(O)/C(NC([C@@H]1C(C)(C)C1)=O)=C/CCCCSC[C@H](N)C(O[Na])=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Cilastatin sodium (MK0791 sodium) 是一种可逆的竞争性的肾脏脱氢肽酶 I (renal dehydropeptidase I) 抑制剂,IC50为 0.1 μM。Cilastatin sodium 抑制细菌金属叶内酰胺酶CphA的IC50为 178 μM。Cilastatin sodium 可用作抗菌辅助剂。 |
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