Pristimerin
Cat. No.:YN251566
CAS No. :1258-84-0
产品名称: | Pristimerin |
CAS No.: | 1258-84-0 |
Chemical Name: | 3-hydroxy-9β,13α-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid, methyl ester |
Synonyms: | Celastrol methyl ester |
分子量: | 464.64 |
分子式: | C₃₀H₄₀O₄ |
SMILES: | C[C@](C1=CC=C(C(C)=C2O)C3=CC2=O)(CC[C@]4(C)[C@@]5([H])C[C@@](C(OC)=O)(C)CC4)[C@]5(CC[C@]13C)C |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Pristimerin是高效可逆的单酰基甘油脂肪酶(MGL)抑制剂,IC50值为93 nM。 |
IC50和靶点: | |
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Solvent & Solubility: |
King, A.R., Dotsey, E.Y., Lodola, A., et al.Discovery of potent and reversible monoacylglycerol lipase inhibitorsChem. Biol.16(10),1045-1052(2009)