ELN-441958
Cat. No.：YN320943
CAS No. ：913064-47-8
| 产品名称: | ELN-441958 |
| CAS No.: | 913064-47-8 |
| Chemical Name: | |
| Synonyms: | ELN 441958 |
| 分子量: | 501.02 |
| 分子式: | C₂₉H₂₉ClN₄O₂ |
| SMILES: | ClC1=C2C(CN(C3=CC=CC(C(N4CCC5(CCN(C6=CC=NC=C6)CC5)CC4)=O)=C3)C2=O)=CC=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | ELN-441958是有效的B1受体拮抗剂, 抑制B1激动剂配体[3H] DAKD与IMR-90细胞结合, Ki值为 0.26 nM, ELN-441958抑制B1受体比作抑制 B2受体具有更高的选择性, 比抑制μ/δ阿片受体选择性分别高500和2000多倍。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
