[Des-Arg9]-Bradykinin
Cat. No.:YN321831
产品名称: | [Des-Arg9]-Bradykinin |
CAS No.: | 15958-92-6 |
Chemical Name: | 1-8-bradykinin |
Synonyms: | [Des-Arg9]-缓激肽 |
分子量: | 904.02 |
分子式: | C₄₄H₆₁N₁₁O₁₀ |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | [Des-Arg9]-Bradykinin 是一种Bradykinin(B1) 受体激动剂,对 B1受体选择性比B2受体高。 |
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Bastian, S., Loillier, B., Paquet, J.L., et al.Stable expression of human kinin B1 receptor in 293 cells: Pharmacological and functional characterizationBr. J. Pharmacol.122(2),393-399(1997)
Leeb-Lundberg, L.M.F., Marceau, F., Müller-Esterl, W., et al.International union of pharmacology. XLV. Classification of the kinin receptor family: From molecular mechanisms to pathophysiological consequencesPharmacol. Rev.57(1),27-77(2005)
Hess, J.F., Borkowski, J.A., Macneil, T., et al.Differential pharmacology of cloned human and mouse B2 bradykinin receptorsMol. Pharmacol.45(1),1-8(1994)
Rhaleb, N.E., Drapeau, G., Dion, S., et al.Structure-activity studies on bradykinin and related peptides: AgonistsBr. J. Pharmacol.99(3),445-448(1990)
Drapeau, G., deBlois, D., and Marceau, F.Hypotensive effects of Lys-des-Arg9-bradykinin and metabolically protected agonists of B1 receptors for kininsJ. Pharmacol. Exp. Ther.259(3),997-1003(1991)