CDK12-IN-E9
Cat. No.:YN290154
CAS No. :2020052-55-3
产品名称: | CDK12-IN-E9 |
CAS No.: | 2020052-55-3 |
Chemical Name: | |
Synonyms: | E9;CDK12-IN-E9 |
分子量: | 434.53 |
分子式: | C₂₄H₃₀N₆O₂ |
SMILES: | C=CC(NC1=CC=CC(NC2=CC(N3[C@H](CCO)CCCC3)=NC4=C(CC)C=NN24)=C1)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CDK12-IN-E9 是一种有效的选择性共价CDK12抑制剂和非共价CDK9抑制剂,同时避免了 ABC 转运蛋白介导的外排。CDK12-IN-E9 对 CDK7/CyclinH 复合物的结合能力较弱,IC50> 1 μM。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |