PD173212
Cat. No.：YN360132
| 产品名称: | PD173212 |
| CAS No.: | 217171-01-2 |
| Chemical Name: | N-[[4-(1,1-dimethylethyl)phenyl]methyl]-N-methyl-L-leucyl-N-(1,1-dimethylethyl)-O-(phenylmethyl)-L-tyrosinamide |
| Synonyms: | Compound 11 |
| 分子量: | 599.85 |
| 分子式: | C₃₈H₅₃N₃O₃ |
| SMILES: | O=C(NC(C)(C)C)[C@@H](NC([C@H](CC(C)C)N(C)CC1=CC=C(C(C)(C)C)C=C1)=O)CC2=CC=C(OCC3=CC=CC=C3)C=C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PD173212 是一种 N-型电压敏感性钙通道 (N-type voltage sensitive calcium channel) 阻滞剂，在 IMR-32 实验中，IC50值为 36 nM。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
Hu, L.-Y., Ryder, T.R., Rafferty, M.F., et al.Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockersBioorg. Med. Chem. Lett.9(15),2151-2156(1999)
