EHP-101
Cat. No.:YN320662
产品名称: | EHP-101 |
CAS No.: | 1818428-24-8 |
Chemical Name: | |
Synonyms: | VCE-004.8 |
分子量: | 433.58 |
分子式: | C₂₈H₃₅NO₃ |
SMILES: | O=C1C(O)=C([C@@H]2C=C(C)CC[C@H]2C(C)=C)C(C(NCC3=CC=CC=C3)=C1CCCCC)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | EHP-101 (VCE-004.8) 是一种口服有效的,特异性PPARγ和CB2受体双重激动剂。EHP-101 可以抑制脯氨酰-羟化酶 (PHDs) 并激活HIF通路。EHP-101 是半合成,多靶点大麻喹啉,具有有效的抗炎活性。EHP-101 减弱脂肪生成并防止饮食诱导的肥胖。 |
IC50和靶点: | |
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In Vivo: | |
Clinical Trial: | |
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