O-2050
Cat. No.:YN320728
产品名称: | O-2050 |
CAS No.: | 1883545-42-3 |
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分子量: | 417.56 |
分子式: | C₂₃H₃₁NO₄S |
SMILES: | CS(=O)(NCCCC#CCC1=CC(O)=C([C@@]2([H])[C@](CC=C(C)C2)([H])C(C)(C)O3)C3=C1)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | O-2050 is a high affinitycannabinoid CB1receptorsilent antagonist. O-2050 also acts as a partial agonist in inhibiting forksolin-induced cyclic AMP stimulation (EC50=40.4 nM). O-2050 antagonizes effects of CP-55940 in vitro. |
IC50和靶点: | [{name:"CB1:2.5 nM (Ki)"},{name: "CB2:0.2 nM (Ki)"}] |
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