AM281
Cat. No.：YN320740
CAS No. ：202463-68-1
| 产品名称: | AM281 |
| CAS No.: | 202463-68-1 |
| Chemical Name: | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-4-morpholinyl-1H-pyrazole-3-carboxamide |
| Synonyms: | 1-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-4-吗啉基-1H-吡唑-3-甲酰胺 |
| 分子量: | 557.21 |
| 分子式: | C₂₁H₁₉Cl₂IN₄O₂ |
| SMILES: | O=C(C1=NN(C2=CC=C(Cl)C=C2Cl)C(C3=CC=C(I)C=C3)=C1C)NN4CCOCC4 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | AM281 是一种选择性CB1受体拮抗剂，IC50为 9.91 nM。AM281 抑制 CB2 受体，IC50为 13000 nM。 |
| IC50和靶点: | [{name:"CB1:9.91 nM (IC50)"},{name: "CB2:13000 nM (IC50)"}] |
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| Solvent & Solubility: |
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