Yangonin
Cat. No.:YN321736
产品名称: | Yangonin |
CAS No.: | 500-62-9 |
Chemical Name: | 4-methoxy-6-[(1E)-2-(4-methoxyphenyl)ethenyl]-2H-pyran-2-one |
Synonyms: | 甲氧醉椒素 |
分子量: | 258.27 |
分子式: | C₁₅H₁₄O₄ |
SMILES: | O=C1C=C(OC)C=C(/C=C/C2=CC=C(OC)C=C2)O1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Yangonin 对人重组大麻素CB1受体具有高的亲和力,IC50和Ki分别为 1.79 μM 和 0.72 μM。 |
IC50和靶点: | [{name:"CB1:1.79 μM (IC50)"},{name: "CB1:0.72 μM (Ki)'}, 'RelA'] |
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Solvent & Solubility: |
Ligresti, A., Villano, R., Allará, M., et al.Kavalactones and the endocannabinoid system: The plant-derived yangonin is a novel CB1 receptor ligandPharmacol. Res.66(2),163-169(2012)