Sograzepide
Cat. No.：YN320919
CAS No. ：155488-25-8
| 产品名称: | Sograzepide |
| CAS No.: | 155488-25-8 |
| Chemical Name: | |
| Synonyms: | Netazepide; YF 476; YM-220 |
| 分子量: | 498.58 |
| 分子式: | C₂₈H₃₀N₆O₃ |
| SMILES: | O=C(NC1=CC=CC(NC)=C1)N[C@H]2C(N(CC(C(C)(C)C)=O)C3=CC=CC=C3C(C4=NC=CC=C4)=N2)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Sograzepide (Netazepide; YF 476; YM-220) 是一种非常有效，高选择性和口服活性的Gastrin/CCK-B拮抗剂，IC50值为 0.1 nM，还抑制Gastrin/CCK-A活性，IC50值_x000D_ 为 502 nM。Sograzepide (Netazepide; YF 476; YM-220) 取代 [125I]CCK-8 与大鼠脑，克隆犬和人Gastrin/CCK-B的特异性结合，Ki值分别为 0.068、0.62 和 0.19 nM。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
