GSK-626616
Cat. No.：YN440105
CAS No. ：1025821-33-3
规格
价格(RMB)
库存
| 产品名称: | GSK-626616 |
| CAS No.: | 1025821-33-3 |
| Chemical Name: | (5Z)-2-[(2,6-dichlorophenyl)amino]-5-(6-quinoxalinylmethylene)-4(5H)-thiazolone |
| Synonyms: | |
| 分子量: | 401.27 |
| 分子式: | C₁₈H₁₀Cl₂N₄OS |
| SMILES: | O=C1N=C(NC2=C(Cl)C=CC=C2Cl)S/C1=C\C3=CC=C4N=CC=NC4=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | GSK-626616 是一种有效的口服生物可利用的DYRK3抑制剂，IC50为 0.7 nM。GSK-626616 以相似的效力抑制 DYRK 家族的其他成员 (例如，DYRK1A和DYRK2)，GSK-626616 可用于贫血研究。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
Erickson-Miller, C.L., Creasy, C., Chadderton, A., et al.GSK626616: A DYRK3 inhibitor as a potential new therapy for the treatment of anemia.Blood110(11),510(2007)
