CLK-IN-T3
Cat. No.:YN440169
产品名称: | CLK-IN-T3 |
CAS No.: | 2109805-56-1 |
Chemical Name: | |
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分子量: | 482.58 |
分子式: | C₂₈H₃₀N₆O₂ |
SMILES: | CC(C1=CC=C(C(NC2=CN3C=C(C4=CC=NC=C4)C=CC3=N2)=O)C=C1)(C)C(N5CCN(C)CC5)=O |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CLK-IN-T3 是一种高效,选择性和稳定的 CDC 样激酶(CLK)抑制剂,对 CLK1,CLK2 和 CLK3 蛋白激酶的IC50分别为 0.67 nM,15 nM 和 110 nM。CLK-IN-T3 具有抗癌活性。 |
IC50和靶点: | [{name:"CLK1:0.67 nM (IC50)"},{name: "CLK2:15 nM (IC50)"},{name: "CLK3:110 nM (IC50)"},{name: "DYRK1A:260 nM (IC50)"},{name: "DYRK1B:230 nM (IC50)"}] |
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