Raclopride
Cat. No.：YN1730019
CAS No. ：84225-95-6
| 产品名称: | Raclopride |
| CAS No.: | 84225-95-6 |
| Chemical Name: | 3,5-dichloro-N-[[(2S)-1-ethyl-2-pyrrolidinyl]methyl]-2-hydroxy-6-methoxy-benzamide |
| Synonyms: | 雷氯必利 |
| 分子量: | 347.24 |
| 分子式: | C₁₅H₂₀Cl₂N₂O₃ |
| SMILES: | O=C(NC[C@H]1N(CC)CCC1)C2=C(OC)C(Cl)=CC(Cl)=C2O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Raclopride 是一种多巴胺D2/D3受体拮抗剂，结合到D2和D3受体，Ki分别为 1.8 nM 和 3.5 nM，但对 D1和 D4受体的亲和力非常低，Ki分别为 18000 nM 和 2400 nM。 |
| IC50和靶点: | [{name:"D2 Receptor:1.8 nM (Ki)"},{name: "D3 Receptor:3.5 nM (Ki)"},{name: "D4 Receptor:2400 nM (Ki)"},{name: "D1 Receptor:18000 nM (Ki)"}] |
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| Solvent & Solubility: |
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