SKF-82958 hydrobromide
Cat. No.：YN1730021
CAS No. ：74115-01-8
| 产品名称: | SKF-82958 hydrobromide |
| CAS No.: | 74115-01-8 |
| Chemical Name: | 6-chloro-2,3,4,5-tetrahydro-1-phenyl-3-(2-propen-1-yl)-1H-3-benzazepine-7,8-diol, monohydrobromide |
| Synonyms: | (±)-SKF 82958 hydrobromide;Chloro-APB hydrobromide |
| 分子量: | 410.73 |
| 分子式: | C₁₉H₂₁BrClNO₂ |
| SMILES: | OC1=C(O)C=C2C(C3=CC=CC=C3)CN(CC=C)CCC2=C1Cl.[H]Br |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | SKF-82958 ((±)-SKF 82958) hydrobromide 是多巴胺D1受体激动剂 (K0.5=4 nM)，对 D1 受体有选择性(K0.5=73 nM)。SKF-82958 hydrobromide 诱导大鼠纹状体膜多巴胺 D1 受体依赖性腺苷酸环化酶活性(EC50=491 nM)。 |
| IC50和靶点: | |
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