LDN-212320
Cat. No.：YN360371
CAS No. ：894002-50-7
| 产品名称: | LDN-212320 |
| CAS No.: | 894002-50-7 |
| Chemical Name: | 3-[[(2-methylphenyl)methyl]thio]-6-(2-pyridinyl)-pyridazine |
| Synonyms: | LDN-0212320; OSU-0212320 |
| 分子量: | 293.39 |
| 分子式: | C₁₇H₁₅N₃S |
| SMILES: | CC1=CC=CC=C1CSC2=NN=C(C3=NC=CC=C3)C=C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | LDN-212320 (LDN-0212320) 是谷氨酸转运体(GLT-1)/兴奋性氨基酸转运体 2(EAAT2)的激活剂。LDN-212320 (LDN-0212320) 通过上调海马和 ACC 星形胶质细胞 GLT-1 的水平来预防伤害性疼痛。 |
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| Solvent & Solubility: |
Kong, Q., Chang, L.-C., Takahashi, K., et al.Small-molecule activator of glutamate transporter EAAT2 translation provides neuroprotectionJ. Clin. Invest.124(3),1255-1267(2014)
