GW311616 hydrochloride
Cat. No.:YN372362
产品名称: | GW311616 hydrochloride |
CAS No.: | 197890-44-1 |
Chemical Name: | (3S,3aS,6aR)-hexahydro-3-(1-methylethyl)-1-(methylsulfonyl)-4-[(2E)-1-oxo-4-(1-piperidinyl)-2-buten-1-yl]-pyrrolo[3,2-b]pyrrol-2(1H)-one, monohydrochloride |
Synonyms: | GW311616A |
分子量: | 433.99 |
分子式: | C₁₉H₃₂ClN₃O₄S |
SMILES: | O=C1[C@@H](C(C)C)[C@@](N(C(/C=C/CN2CCCCC2)=O)CC3)([H])[C@]3([H])N1S(=O)(C)=O.[H]Cl |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | GW-311616 是高活性,口服生物相容性,长效的人中性白细胞弹性蛋白酶 (HNE) 抑制剂,IC50为 22 nM,Ki为 0.31 nM。 |
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